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Tuneable access to indole, indolone and cinnoline derivatives from a common 1,4-diketone Michael acceptor

Article scientifique 2020 Anglais

Résumé

A convergent strategy is reported for the construction of nitrogen-containing heterocycles from common substrates: 1,4-diketones and primary amines. Indeed, by just varying substrates, substituents or heating mode it is possible to selectively synthesize indole, indolone (1,5,6,7-tetradihydroindol-4-one) or cinnoline (5,6,7,8-tetrahydrocinnoline) derivatives in moderate to excellent yields.

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El-Marrouki, D., Touchet, S., Abdelli, A., M’rabet, H., Efrit, M., Gros, P. (2020). Tuneable access to indole, indolone and cinnoline derivatives from a common 1,4-diketone Michael acceptor. https://doi.org/10.3762/bxiv.2020.56.v1

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Auteur(s)

Dalel El-Marrouki Sabrina Touchet Abderrahmen Abdelli Hédi M’rabet Mohamed Lotfi Efrit Philippe C. Gros

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